Medicines play a vital role in the rehabilitation process following sports injuries, aiding in pain management, reducing inflammation, and promoting faster recovery. This article provides a comprehensive overview of the chemistry of drugs commonly used in sports medicine, including their synthesis, molecular structures, and practical applications. In addition, the discussion includes an analysis of the current market trends and demand for these pharmaceutical agents, providing insight into their commercial relevance. Special emphasis is placed on analgesics and anti-inflammatory drugs, which are essential for the immediate therapeutic treatment of injuries sustained during sports activities. These medications not only help alleviate pain but also control inflammation, enabling athletes to recover more efficiently and safely. Overall, the article aims to bridge the understanding of both the chemical and clinical aspects of these drugs in the context of sports injury management.